Chemren Bio-Engineering Co., Ltd.

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Product name : 4SC-202
Item : CR2029
CAS : 1186222-89-8
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Details:

Biological Activity of 4SC-202

4SC-202 is an orally available potent HDACi specific for class I HDAC isoenzymes(NO HDAC8) with IC50s of 1.2/1.12/0.57 uM for HDAC1/2/3; high selectivity over ClassIIa/IIb/III HDACs.
IC50 value:
Target: HDAC1/2/3
The novel HDACi 4SC-202 is an orally available potent HDACi specific for class I HDAC isoenzymes. It has shown substantial anti-tumour activity in a broad panel of cancer cell lines as well as in various cancer xenograft models. A Phase I study with 4SC-202 in haematological malignancies is currently prepared and about to start soon

Chemical Information

M.Wt 619.71 Storage Please store the product under the recommended conditions in the Certificate of Analysis.
Formula C30H29N5O6S2
CAS No 1186222-89-8
Solvent & Solubility

DMSO 50 mg/ml

Preparing Stock Solutions

1 mg 5 mg 10 mg
1 mM 1.6137 mL 8.0683 mL 16.1366 mL
5 mM 0.3227 mL 1.6137 mL 3.2273 mL
10 mM 0.1614 mL 0.8068 mL 1.6137 mL

References on 4SC-202

Availability and price:
Stock : in stock
We offer significant discount for larger quantity order.
For quotation, question, and order, please send email to :sales@chemrenpharm.com

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